Development of Osmotically Controlled Mucoadhesive Cup-Core (OCMC) Tablet for The Anti-Inflammatory Activity

AuthorHitesh Ranchhodbhai Patelen
AuthorMadhabhai Manordas Patelen
Issued Date2010-01-31en
AbstractThe aim of the present study was to prepare and evaluate an osmotically controlled mucoadhesive cup-core (OCMC) containing aceclofenac. A special technique was used while preparing an OCMC. Stability of OCMC was determined in natural human saliva, and it was found that both pH and device are stable in human saliva. OCMC was evaluated by weight uniformity, thickness, hardness, friability, swelling, mucoadhesive strength and in vitro drug release. Swelling index was higher with formulations containing hydroxypropyl methylcellulose (HPMC) K4M alone, and it decreases with its decreasing concentration in the OCMC. The in vitro drug release studies showed a release with the composition of formulation up to 12 h. The mechanism of drug release was found to be zero order kinetics with diffusion controlled drug release. It has shown significant anti-inflammatory activity (Pen
DOIhttps://doi.org/10.22037/ijpr.2010.831en
URIhttps://brieflands.com/journals/ijpr/articles/126034en
KeywordOsmotic cup-core tableten
KeywordAceclofenacen
KeywordMucoadhesionen
KeywordDrug releaseen
KeywordAnti- inflammatory activityen
PublisherBrieflandsen
TitleDevelopment of Osmotically Controlled Mucoadhesive Cup-Core (OCMC) Tablet for The Anti-Inflammatory Activityen
TypeOriginal Articleen

Files

Original bundle

Now showing 1 - 1 of 1
Loading...
Thumbnail Image
Name:
ijpr-09-21.pdf
Size:
546.91 KB
Format:
Adobe Portable Document Format
Description:
Article/s PDF